Inhibitor

GnRH Associated Peptide (GAP) (1-13), human | A1020-10 | Gentaur US, UK & Europe Disrtribition Purity: 0.9941 Short Sumary: Inhibitor of prolactin secretion Category: Endocrinology and...

GnRH Associated Peptide (GAP) (1-13), human | A1020-1 | Gentaur US, UK & Europe Disrtribition Purity: 0.9941 Short Sumary: Inhibitor of prolactin secretion Category: Endocrinology and...

GnRH Associated Peptide (GAP) (1-13), human | A1020-5 | Gentaur US, UK & Europe Disrtribition Purity: 0.9941 Short Sumary: Inhibitor of prolactin secretion Category: Endocrinology and...

Glucagon (19-29), human | A1019-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.9554 Short Sumary: Potent Ca2+/Mg2+-ATPase inhibitor Category: Endocrinology and Hormones#Obesity#...

Glucagon (19-29), human | A1019-10 | Gentaur US, UK & Europe Disrtribition Purity: 0.9554 Short Sumary: Potent Ca2+/Mg2+-ATPase inhibitor Category: Endocrinology and Hormones#Obesity#...

Glucagon (19-29), human | A1019-5 | Gentaur US, UK & Europe Disrtribition Purity: 0.9554 Short Sumary: Potent Ca2+/Mg2+-ATPase inhibitor Category: Endocrinology and Hormones#Obesity#...

Anti-Inflammatory Peptide 1 | A1008-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.9999 Short Sumary: PLA2 inhibitor Category: Immunology/Inflammation Synonyms: ...

Anti-Inflammatory Peptide 1 | A1008-10 | Gentaur US, UK & Europe Disrtribition Purity: 0.9999 Short Sumary: PLA2 inhibitor Category: Immunology/Inflammation Synonyms: ...

Anti-Inflammatory Peptide 1 | A1008-5 | Gentaur US, UK & Europe Disrtribition Purity: 0.9999 Short Sumary: PLA2 inhibitor Category: Immunology/Inflammation Synonyms: ...

Tankyrase Inhibitors (TNKS) 49 | 27659 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Tankyrase 1 and tankyrase 2 are members of...

Tankyrase Inhibitors (TNKS) 22 | 27658 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Tankyrase 1 and tankyrase 2 are members of...

Tenovin-6 | 27661-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Tenovin-6 is the water soluble...

SMER3 | 27718-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for the inhibition of SCFMET30 in cell-based or in vitro assays. ...

AG-14361 | 27602-3 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: A 17-hour exposure of A549 cells to 0.4 µM AG14361 does not...

Milrinone | 27309 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: PDE InhibitorOur Inhibitors are...

GSK256066 | 27751-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: GSK256066 is a selective PDE4...

Pimobendan | 27638-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Pimobendan is a selective...

Apremilast (CC-10004) | 27735-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Apremilast, also...

RGFP966 | 27643-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: RGFP966 is a slow-on/slow-off, competitive tight-binding...

PCI 34051 | 27317 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Caspase and HDAC Inhibitor Product...

KY 02111 | 27759-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: N/A Description: Promotes differentiation of human ESCs and...

BMN-673 8R,9S | 27610-2 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: BMN-673 is an orally bioavailable inhibitor of the nuclear...

LAQ824 (NVP-LAQ824,Dacinostat) | 27760-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: A recent study shows that LAQ824...

ICG 001 | 27752-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: ICG001 selectively inhibits colon carcinoma cell lines (SW480...

EPZ5676 | 27625-2 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: EPZ5676 is a potent inhibitor of DOT1L histone...

AR-42 (OSU-HDAC42) | 27603-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: AR-42 induces histone H3 acetylation,...

A-966492 | 27601-3 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: A-966492 is one of the most potent PARP inhibitors. A-966492...

CUDC-907 | 27616-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: CUDC-907 has a long half-life in murine tumors. CUDC-907...

BMN 673 | 27609-2 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: BMN673 has shown anti-tumor activity both in vitro and in vivo...

Pracinostat (SB939) | 27771-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Pracinostat (SB939) is an orally...

Caspase-3/7 Inhibitor I | 27741-3 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Selectivity for caspases-3 and 7 involves unique...

(-)-JQ1 | 27335 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: (-)-JQ1 is the inactive stereoisomer of the potent,...

CHIR-99021 (CT99021) HCl | 27615-3 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: Hydrochloride salt of CHIR...

CHIR-99021 (CT99021) | 27614-3 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: CHIR-99021 is a highly specific...

Trimidox | 27320 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis/Inhibitors & Activators Application: N/A Background: N/A Description: Caspase Activator Product Type: ...

Wnt-C59 | 27780-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: Wnt-C59 prevents palmitoylation of Wnt proteins by Porcupine (a...

Z-VEID-FMK | 27669-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: VEID is the specific recognition sequence for caspase-6/Mch2. Caspase...

Z-VDVAD-FMK | 27668-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: VDVAD has been shown to be a preferred cleavage site for caspase-2...

3-Deazaneplanocin A (DZNep) hydrochloride | 27618-2 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: 3-Deazaneplanocin...

3-Deazaneplanocin (DZNep) | 27617-2 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: 3-Deazaneplanocin A (DZNep) is an...

Boc-D-FMK | 27611-3 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Boc-D-FMK is a cell-permeable broad-spectrum caspase inhibitor that...

OTX-015 | 27636-3 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the targeting of...

Oxyresveratrol | 27318 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis/Inhibitors & Activators Application: N/A Background: N/A Description: Caspase-3 Inhibitor Product...

Tenovin-6 | 27661-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Tenovin-6 is the water soluble...

Cilomilast | 27742-3 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Cilomilast, also known as...

TCID | 27720-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for cell-based and in vitro studies of UCH-L3 function. Background:...

Tadalafil | 27657-3 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Tadalafil is a small-molecule inhibitor of...

SGC-CBP30 | 27650-2 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: CREBBP (CBP) and EP300 are general transcriptional...

Q-VD(OMe)-OPh | 27640-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Q-VD-OPh is a broad spectrum caspase inhibitor that provides a cost...

CAY10625 | 27321 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis/Inhibitors & Activators Application: N/A Background: N/A Description: Caspase-3 and -7 Inhibitor Product...

XL-888 | 27781-3 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: X-ray crystallographic analysis reveals that the...

PYR-41 | 27716-3 | Gentaur US, UK & Europe Disrtribition Category: Protease/Inhibitors / Activators Application: Useful for inhibition of E1 ubiquitin conjugating enzymes Background: N/A ...

PR-619 | 27714-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for non-specific inhibition of ubiquitin-like isopeptidases for...

PS-341 (MG-341) | 27715-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for as a potent, cell permeable proteasome inhibitor for...

PCI 34051 | 27316 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Caspase and HDAC Inhibitor Product...

NU 7026 | 27312 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: PARP3 Inhibitor Product Type: Inhibitor ...

Milrinone | 27308 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: PDE Inhibitor Product Type: ...

VX-765 | 27779-1 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: VX-765 is an orally-absorbed pro-drug of VRT-043198, a potent and...

NVP-BEP800 | 27766-3 | Gentaur US, UK & Europe Disrtribition Category: Protease/Inhibitors / Activators Application: N/A Background: NVP-BEP800 binds to the N-terminal ATP-binding pocket of...

SGI-1776 free base | 27651-3 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: According to preliminary results from studies treating...

Posaconazole | 27639-2 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: Posaconazole, also known as SCH 56592 or Noxafil, is...

OG-L002 | 27635-2 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: N/A Description: N/A Product Type: Inhibitor ...

Z-FA-FMK | 27667-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: N/A Description: N/A Product Type: Inhibitor Shippement...

Z-DQMD-FMK | 27666-3 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Z-DQMD-FMK is a potent cell-permeable inhibitor of caspase-3...

C646 | 27613-2 | Gentaur US, UK & Europe Disrtribition Category: Acetyltransferase/Inhibitors / Activators Application: N/A Background: C646 binds to p300 as the Z-isomer forming hydrogen...

PCI-24781 (CRA-024781) | 27769-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: PCI-24781 is a pan-HDAC inhibitor that...

P22077 | 27712-2 | Gentaur US, UK & Europe Disrtribition Category: Protease/Inhibitors / Activators Application: Useful for inhibition of USP7 and USP47 activity. Background: N/A ...

Roflumilast | 27645-3 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: The enzyme PDE-4 is found mainly in...

JNJ-26481585 | 27632-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Quisinostat, also known asJNJ-26481585, is an orally...

SB 939 | 27331 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: HDAC Inhibitor Product Type: ...

EPZ015666 | 79043-2 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: N/A Description: EPZ015666 is a potent,...

Oxamflatin | 27326 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: HDAC Inhibitor Product Type: ...

Z-VAD(OMe)-FMK | 27313 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: N/A Description: Z-VAD(OMe)-FMK is a cell permeable, irreversible...

Vardenafil HCl Trihydrate | 27776-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Vardenafil is frequently used in...

Rucaparib (AG-014699,PF-01367338) | 27647-3 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Rucaparib, also named as AG-014699 or...

Belinostat (PXD101) | 27608-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Belinostat has been found to significantly...

Embelin | 27322 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis/Inhibitors & Activators Application: N/A Background: N/A Description: XIAP Inhibitor Product Type: Inhibitor...

LDN-57444 | 27706-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for the inhibition of Ubiquitin C-terminal Hydrolase (UCH-L1) in...

Celastrol | 27702-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for inhibition of NF-κappa-B-dependent pathways and inhibition...

Caspase-3/7 Inhibitor I | 27741-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Selectivity for caspases-3 and 7 involves unique...

EPZ-6438 | 27626-3 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: EPZ-6438 competitively binds to the...

3-Deazaneplanocin A (DZNep) hydrochloride | 27618-1 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: 3-Deazaneplanocin...

3-Deazaneplanocin (DZNep) | 27617-1 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: 3-Deazaneplanocin A (DZNep) is an...

GSK J4 HCl | 27627-2 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: GSK J4 is a potent cell-permeable inhibitor of the...

Z-FA-FMK | 27667-3 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: N/A Description: N/A Product Type: Inhibitor Shippement...

I-BET151 (GSK1210151A) | 27629-3 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the...

Apoptosis Inhibitor | 27734-3 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: N/A Description: Apoptosis Inhibitor is a cell-permeable...

OTX-015 | 27636-2 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the targeting of...

Trimidox | 27319 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis/Inhibitors & Activators Application: N/A Background: N/A Description: Caspase Activator Product Type: ...

IPI-504 (Retaspimycin hydrochloride) | 27753-1 | Gentaur US, UK & Europe Disrtribition Category: Protease/Inhibitors / Activators Application: N/A Background: Cancer cells depend on the...

Telotristat | 27341 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: N/A Description: Telotristat is the active...

SIRT1/2 Inhibitor IV | 27323 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: SIRT1/2 Inhibitor...

IWP-L6 | 27755-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: WP-L6 was developed as a sub-nanomolar inhibitor of Porcupine,...

Tenovin-1 | 27660-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Tenovin-1, a small molecule discovered by a cell-based...

S- (+)-Rolipram | 27648-3 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Rolipram is a racemic drug that increases...

ME0328 | 27634-2 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: ME0328 is a potent and selective PARP...

ML161 | 27764-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: ML-161 is thought to act allosterically. ML-161 inhibits...

Romidepsin (FK228, depsipeptide) | 27646-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Romidepsin is a bicyclic...

I-BET-762 | 27630-2 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the targeting of...

BMN 673 | 27609-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: BMN673 has shown anti-tumor activity both in vitro and in vivo...