Inhibitor

DBeQ | 27703-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for the study of the ubiquitin-dependent and endoplasmic reticulum-associated degradation pathway (p97 ATPase) Background:...

b-AP15 (NSC-687852) | 27701-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Suitable for validation studies of the deubiquitinating activities of the 19S regulatory particle as a drug target,...

Aminophylline | 27731 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Aminophylline is a bronchodilator that is used together with other medicines to treat the acute...

MC1568 | 27761-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: MC1568, a derivative of (Aryloxopropenyl)pyrrolyl hydroxyamide, is a novel, potent and specific inhibitor of...

Ezetimibe | 27749-3 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: Ezetimibe has been reported to be a cholesterol transport inhibitor. Mechanistic studies show that this...

Tenovin-6 | 27661-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Tenovin-6 is the water soluble analog of Tenovin-1 and acts as a potent SIRT1 and SIRT2...

Rucaparib (AG-014699,PF-01367338) | 27647-2 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Rucaparib, also named as AG-014699 or PF-01367338, is a poly (ADP ribose) polymerase (PARP)...

Romidepsin (FK228, depsipeptide) | 27646-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Romidepsin is a bicyclic depsipeptide antibiotic isolated from the bacterium...

EPZ-6438 | 27626-1 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: EPZ-6438 competitively binds to the S-adenosylmethionine (SAM) binding site of EZH2 and also...

AR-42 (OSU-HDAC42) | 27603-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: AR-42 induces histone H3 acetylation, α-tubulin acetylation and p21 up-regulation, which have been...

Bromosporine | 27612 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the targeting of chromatin-modifying enzymes to specific sites,...

UNC1215 | 27406 | Gentaur US, UK & Europe Disrtribition Category: Methyl-lysine Reader/Inhibitors / Activators Application: N/A Background: N/A Description: UNC 1215 is a methyl-lysine inhibitor. UNC1215 inhibits L3MBTL3 with 50x more potency...

VX-765 | 27779-2 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: VX-765 is an orally-absorbed pro-drug of VRT-043198, a potent and selective inhibitor of ICE/caspase-1 sub-family caspases...

Pracinostat (SB939) | 27771-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Pracinostat (SB939) is an orally bioavailable, small-molecule histone deacetylase (HDAC) inhibitor...

UNC669 | 27664-2 | Gentaur US, UK & Europe Disrtribition Category: Methyl-lysine Reader/Inhibitors / Activators Application: N/A Background: N/A Description: UNC669 is a potent and selective MBT (malignant brain tumor) inhibitor for L3MBTL1. ...

I-BET151 (GSK1210151A) | 27629-1 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: Bromodomains have an important role in the targeting of chromatin-modifying enzymes to specific...

(-)-JQ1 | 27334 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: (-)-JQ1 is the inactive stereoisomer of the potent, cell-permeable, small molecule bromodomain inhibitor (+)-JQ1...

Cilostazol | 27743-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Cilostazol (OPC-13013, Pletal) is a 2-oxo-quinoline derivative with antithrombotic, vasodilator,...

NSC-632839 | 27709-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for non-specific inhibition of ubiquitin-like isopeptidases for cell biology and drug discovery studies. ...

Tadalafil | 27657-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Tadalafil is a small-molecule inhibitor of phosphodiesterase 5 (PDE5), a predominant PDE in the...

Roflumilast | 27645-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: The enzyme PDE-4 is found mainly in inflammatory cells, and Roflumilast acts as a selective,...

JW 55 | 27633-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Inhibitor of the PARP domain of tankyrase 1 and 2 (TNKS1/2). Activity results in stabilization of Axin2 and increased...

Wnt-C59 | 27780-3 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: Wnt-C59 prevents palmitoylation of Wnt proteins by Porcupine (a membrane-bound O-acyltransferase), thereby blocking...

PCI-24781 (CRA-024781) | 27769-3 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: PCI-24781 is a pan-HDAC inhibitor that shows antitumor activity in vitro and in vivo...

NVP-BEP800 | 27766-2 | Gentaur US, UK & Europe Disrtribition Category: Protease/Inhibitors / Activators Application: N/A Background: NVP-BEP800 binds to the N-terminal ATP-binding pocket of Hsp90. Hsp90 is a ubiquitously expressed molecular...

NSC697923 | 27765-2 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: N/A Background: NSC697923 selectively inhibits PMA-induced NF-?B activation, and also inhibits I?Bα phosphorylation by both...

WP1130 | 27722-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Suitable for cell-based studies of USP function. Background: N/A Description: A partially-selective, cell permeable DUB...

LDN-57444 | 27706-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: Useful for the inhibition of Ubiquitin C-terminal Hydrolase (UCH-L1) in drug discovery studies. Background: N/A ...

Rocilinostat (ACY-1215) | 27644-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Rocilinostat, also known as ACY-1215, is a selective HDAC6 inhibitor with...

VER 155008 | 27777-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: VER 155008 is a potent inhibitor of heat shock protein 70 (Hsp70) family of chaperones, which have been...

ML161 | 27764-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: ML-161 is thought to act allosterically. ML-161 inhibits thrombin-induced platelet activation. Description: ...

ICG 001 | 27752-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: ICG001 selectively inhibits colon carcinoma cell lines (SW480 and HCT-116 cells) but not normal colonic epithelial...

RGFP966 | 27643-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: RGFP966 is a slow-on/slow-off, competitive tight-binding HDAC inhibitor. RGFP966 treatment on two CTCL cell...

GSK J4 HCl | 27627-1 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: GSK J4 is a potent cell-permeable inhibitor of the histone H3 lysine 27 (H3K27) demethylase JMJD3. GSK J4 is...

AZD2461 | 27606-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Unlike treatment with AZD 2281 (Olaparib, Axon 1464), AZD 2461 succesfully circumvents drug resistance of...

A-966492 | 27601-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: A-966492 is one of the most potent PARP inhibitors. A-966492 displays excellent potency against the PARP-1 enzyme with...

ND-630 | 27071-1 | Gentaur US, UK & Europe Disrtribition Category: Metabolic Enzymes/Inhibitors Application: N/A Background: N/A Description: ND-630 (NDI 010976) is a highly specific, reversible inhibitor of ACC1 (IC50 = 2 nM) and ACC2 (IC50...

Tubacin | 27662 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Tubacin is a highly potent and selective, reversible, cell-permeable HDAC6 inhibitor . Tubacin...

Sodium Phenylbutyrate | 27654 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Sodium Phenylbutyrate is a transcriptional regulator that acts by altering...

IWP-L6 | 27755-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: WP-L6 was developed as a sub-nanomolar inhibitor of Porcupine, the enzyme that catalyzes the palmitoylation of Wnt...

Ezetimibe | 27749-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: Ezetimibe has been reported to be a cholesterol transport inhibitor. Mechanistic studies show that this...

Tubastatin A | 27663-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: N/A Product Type: Inhibitor Shippement Condition: Room temp. (continental US) or...

OG-L002 | 27635-1 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: N/A Description: N/A Product Type: Inhibitor Shippement Condition: Room temp. (continental US) or gel...

C646 | 27613-1 | Gentaur US, UK & Europe Disrtribition Category: Acetyltransferase/Inhibitors / Activators Application: N/A Background: C646 binds to p300 as the Z-isomer forming hydrogen bonds between Thr1411, tYR1467, Trp1466 and Arg1410 on...

Levodopa | 79792 | Gentaur US, UK & Europe Disrtribition Category: Neuroscience/Inhibitors Application: N/A Background: N/A Description: Levodopa is a dopamine precursor that is being studied as a potential treatment for the symptoms of...

Carbidopa | 79791 | Gentaur US, UK & Europe Disrtribition Category: Neuroscience/Inhibitors Application: N/A Background: N/A Description: Carbidopa is a decarboxylase inhibitor used in conjunction with levodopa in patients with Parkinson's...

Epacadostat (INCB024360) | 27339-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: Epacadostat (INCB024360) is an orally available hydroxyamidine and...

Epacadostat (INCB024360) | 27339-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: Epacadostat (INCB024360) is an orally available hydroxyamidine and...

INCB024360 Analog | 27338-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: INCB024360 analog is an orally available hydroxyamidine and inhibitor of...

INCB024360 Analog | 27338-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: INCB024360 analog is an orally available hydroxyamidine and inhibitor of...

NLG919 | 27337-2 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: NLG919 is an orally available potent inhibitor of the indoleamine-2,3- dioxygenase (IDO)...

NLG919 | 27337-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Immunotherapy Application: N/A Background: N/A Description: NLG919 is an orally available potent inhibitor of the indoleamine-2,3- dioxygenase (IDO1)...

(+)-JQ1 | 27400 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: N/A Description: (+)-JQ1 is a specific inhibitor of the BET family of acetyl-lysine recognition motifs,...

1,5-Isoquinolinediol | 27310 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: PARP1 Inhibitor Product Type: Inhibitor Shippement Condition: room temp or gel...

Ruxolitinib, Phosphate | 27059-2 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: Ruxolitinib, also known as INCB18424, is a potent and selective Janus kinase JAK1 and...

Ruxolitinib, Phosphate | 27059-1 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: Ruxolitinib, also known as INCB18424, is a potent and selective Janus kinase JAK1 and...

SMI-4a | 27774-1 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: The serine/threonine Pim kinases have been suggested to promote the activity of the rapamycin-sensitive mammalian target of...

Alvespimycin HCl (17-DMAG) | 27730-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Metabolic Enzymes Application: N/A Background: Alvespimycin hydrochloride is the hydrochloride salt of alvespimycin, an analogue of...

Droxinostat | 27620-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Droxinostat has shown a potent action against HDAC3, HDAC6, and HDAC8 which are pyrimidyl-hydroxamic...

Cisplatin | 27744 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: Cisplatin induces cytotoxicity by interaction with DNA to form intrastrand crosslinks which activate several signal transduction...

Vardenafil HCl Trihydrate | 27776-2 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Vardenafil is frequently used in the treatment erectile dysfunction, and is the active...

EPZ005687 | 27624-1 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: EPZ005687 is a potent inhibitor of EZH2, an enzymatic subunit of polycomb repressive complex 2 (PRC2)...

Rolipram | 27005 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Rolipram is a selective, cell permeable inhibitor of cAMP-specific phosphodiesterase 4...

UPF 1069 | 27665-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: UPF 1069, a derivative of isoquinolinone, is a potent and selective inhibitor of poly-(ADP-ribose)...

Tenovin-1 | 27660-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Tenovin-1, a small molecule discovered by a cell-based screen, is a bio-active activator of p53 that elevates...

SGI-1776 free base | 27651-1 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: According to preliminary results from studies treating prostate cancer cells, SGI-1776 dose-dependently reduces...

3-aminobenzamide | 79888-2 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: 3-aminobenzamide can sensitize cells to radiation in vitro by inhibiting the repair of DNA damage,...

Cilomilast | 27742-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Cilomilast, also known as SB-207499 or Ariflo, is a potent second generation...

Apoptosis Inhibitor | 27734-1 | Gentaur US, UK & Europe Disrtribition Category: Apoptosis Inhibitor Application: N/A Background: N/A Description: Apoptosis Inhibitor is a cell-permeable inhibitor of apoptosis induction. It does not directly...

S- (+)-Rolipram | 27648-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Rolipram is a racemic drug that increases brain cAMP availability by inhibiting phosphodiesterase...

PI-103 | 27502-1 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: PI-103 is a multi-targeted inhibitor of PI3K for p110, p110, p110 , and p110 with reported IC50...

P005091 | 27767-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: N/A Background: USP7, known as herpes-associated-ubiquitin-specificprotease (HAUSP), is a deubiquitylating enzyme that...

UNC669 | 27664-1 | Gentaur US, UK & Europe Disrtribition Category: Methyl-lysine Reader/Inhibitors / Activators Application: N/A Background: N/A Description: UNC669 is a potent and selective MBT (malignant brain tumor) inhibitor for L3MBTL1. ...

Rocilinostat (ACY-1215) | 27644-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Rocilinostat, also known as ACY-1215, is a selective HDAC6 inhibitor with...

Posaconazole | 27639-1 | Gentaur US, UK & Europe Disrtribition Category: Demethylase/Inhibitors / Activators Application: N/A Background: Posaconazole, also known as SCH 56592 or Noxafil, is a novel triazole antifungal compound that potently...

Donepezil HCl | 27619-1 | Gentaur US, UK & Europe Disrtribition Category: Metabolic Enzymes/Inhibitors Application: N/A Background: Donepezil HCl is a piperidine-class AChE inhibitor containing an N-benzylpiperdine and an indanone moiety, which...

Belinostat (PXD101) | 27608-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Belinostat has been found to significantly increase the acetylation of histones H3 and H4 and exerts...

Vinpocetine | 27778-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: N/A Description: Vinpocetine, also known as Cavinton or ethyl apovincaminate, is a specific...

NSC697923 | 27765-1 | Gentaur US, UK & Europe Disrtribition Category: Ubiquitination/Inhibitors / Activators Application: N/A Background: NSC697923 selectively inhibits PMA-induced NF-?B activation, and also inhibits I?Bα phosphorylation by both...

MC1568 | 27761-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: MC1568, a derivative of (Aryloxopropenyl)pyrrolyl hydroxyamide, is a novel, potent and specific inhibitor of...

Tubastatin A | 27663-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: N/A Product Type: Inhibitor Shippement Condition: Room temp. (continental US) or...

Tadalafil | 27657-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Tadalafil is a small-molecule inhibitor of phosphodiesterase 5 (PDE5), a predominant PDE in the...

Rucaparib (AG-014699,PF-01367338) | 27647-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: Rucaparib, also named as AG-014699 or PF-01367338, is a poly (ADP ribose) polymerase (PARP)...

ME0328 | 27634-1 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: ME0328 is a potent and selective PARP inhibitor with about 7-fold selectivity over PARP3 over PARP1...

Irsogladine | 27754 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Irsogladine is a selective PDE4 inhibitor that facilitates gap junction intercellular communication...

KY 02111 | 27759-1 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: N/A Description: Promotes differentiation of human ESCs and iPSCs into cardiomyocytes. Induces downregulation of...

Kaempferol | 27757 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: N/A Description: Naturally occurring flavonoid found in Gingko biloba and red wines that activates the...

Set of PARP Inhibitors (8 x 50 µl) | 78318 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors Application: N/A Background: N/A Description: A set of Poly (ADP-ribose) polymerases (PARP) inhibitors (PARPi) including PARPi with a...

Novobiocin | 27501 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: N/A Description: Novobiocin is an aminocoumarin antibiotic that is produced by Streptomyces niveus. Along with...

Novo-TRX | 27500 | Gentaur US, UK & Europe Disrtribition Category: Inhibitors / Activators/Other Application: N/A Background: N/A Description: Novobiocin is an aminocoumarin antibiotic that is produced by Streptomyces niveus. Along with other...

RediSolution™ (+)-JQ1 | 27403 | Gentaur US, UK & Europe Disrtribition Category: Bromodomain/Inhibitors / Activators Application: N/A Background: N/A Description: (+)-JQ1 is a specific inhibitor of the BET family of acetyl-lysine recognition...

Sirtinol | 27652-1 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Unlike TSA, Sirtinol does not inhibit class I and class II HDACs, indicating that it is a selective sirtuin...

Dyphylline | 27747 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Dyphylline is a selective A1 and A2 adenosine receptor antagonist. Decreases ABCG2 protein in cells and...

UNC1215 | 27405 | Gentaur US, UK & Europe Disrtribition Category: Methyl-lysine Reader/Inhibitors / Activators Application: N/A Background: N/A Description: UNC 1215 is a methyl-lysine inhibitor. UNC1215 inhibits L3MBTL3 with 50x more potency...

DPQ | 27311 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: PARP1&2 Inhibitor Product Type: Inhibitor Shippement Condition: room temp or gel packs

Parthenolide | 27768-2 | Gentaur US, UK & Europe Disrtribition Category: Deacetylase/Inhibitors / Activators Application: N/A Background: Parthenolide is a sesquiterpene lactone and the active principle of feverfew (Chrysanthemum parthenium) ...

PJ34 | 27041 | Gentaur US, UK & Europe Disrtribition Category: PARP/Inhibitors / Activators Application: N/A Background: N/A Description: A cell-permeable, water-soluble, potent inhibitor of poly(ADP-ribose) polymerase (PARP; EC50 = 20 nM)...

Staurosporine | 27002 | Gentaur US, UK & Europe Disrtribition Category: Kinase/Kinase Inhibitors Application: N/A Background: N/A Description: Staurosporine is a potent inhibitor of many kinases including protein kinase C, protein kinase A,...

Anagrelide HCl | 27732-1 | Gentaur US, UK & Europe Disrtribition Category: Phosphodiesterase/Inhibitors / Activators Application: N/A Background: Anagrelide is a FDA-approved drug for the treatment of essential thrombocythemia. It is originally...

Entacapone | 27621-1 | Gentaur US, UK & Europe Disrtribition Category: Methyltransferase/Inhibitors / Activators Application: N/A Background: N/A Description: Entacapone is a second-generation catechol-O-methyltransferase (COMT) inhibitor...