Receptors

CGP 52432 | B6655-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.9909 Short Sumary: GABAB receptor antagonist Category: Membrane Transporter/Ion Channel|GABA Receptor Synonyms: N/A Formula: C15H24Cl2NO4P N/A Molecular Weight: ...

(2R,4R)-APDC | B6634-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: group II metabotropic glutamate receptor agonist Category: Neuroscience|GluR Synonyms: N/A Formula: C6H10N2O4 N/A Molecular Weight: 174.16 ...

[Sar9,Met (O2)11]-Substance P | B6623-25 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: NK1 tachykinin receptor agonist Category: Neuroscience|Substance P/NK1 Receptor Synonyms: N/A Formula: C64H100N18O15S N/A ...

Senktide | B6580-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: NK3 tachykinin receptor agonist Category: GPCR/G protein|NK3 Receptor Synonyms: N/A Formula: C40H55N7O11S N/A Molecular Weight: 841.97 Chemical...

NBQX disodium salt | B6566-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: A potent, highly selective and competitive AMPA receptor antagonist Category: Membrane Transporter/Ion Channel|AMPAR Synonyms: N/A Formula: ...

(S)-3-Carboxy-4-hydroxyphenylglycine | B6262-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: group I metabotropic glutamate receptor antagonist and group II mGlu agonist Category: Neuroscience|GluR Synonyms: N/A ...

(R)-3-Carboxy-4-hydroxyphenylglycine | B6261-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: NMDA and AMPA/kainate receptor antagonist Category: Neuroscience|GluR Synonyms: N/A Formula: C9H9NO5 N/A Molecular...

(S)-3-Hydroxyphenylglycine | B6260-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: group I metabotropic glutamate receptors agonist Category: Neuroscience|GluR Synonyms: N/A Formula: C8H9NO3 N/A Molecular Weight: ...

(S)-4-Carboxyphenylglycine | B6258-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: group I metabotropic glutamate receptor antagonist Category: Neuroscience|GluR Synonyms: N/A Formula: C9H9NO4 N/A Molecular...

(R)-4-Carboxyphenylglycine | B6257-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: NMDA receptor antagonist Category: Membrane Transporter/Ion Channel|NMDA Receptor Synonyms: N/A Formula: C9H9NO4 N/A Molecular...

(S)-4-Carboxy-3-hydroxyphenylglycine | B6255-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: group I mGlu1a/1a receptor antagonist and mGluR2 agonist Category: Neuroscience|GluR Synonyms: N/A Formula: C9H9NO5 N/A ...

(1S,3R)-ACPD | B6245-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: group I and II mGlu receptor agonist Category: Neuroscience|GluR Synonyms: N/A Formula: C7H11NO4 N/A Molecular Weight: 173.17 Chemical Name: ...

(±)-trans-ACPD | B6220-100 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: metabotropic glutamate receptors agonist Category: Neuroscience|GluR Synonyms: N/A Formula: C7H11NO4 N/A Molecular Weight: 173.17 Chemical...

GSK481 | B6194-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: RIP1 (Receptor Interacting Protein Kinase 1) inhibitor Category: Apoptosis|TNF-α Synonyms: N/A Formula: C21H19N3O4 N/A Molecular Weight: 377.39 ...

ELN441958 | B5925-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Potent and selective bradykinin B1 receptor antagonist Category: GPCR/G protein|Bradykinin Receptors Synonyms: N/A Formula: C29H29ClN4O2 N/A ...

ACT 335827 | B5787-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Orexin receptor 1 antagonist,potent and selective Category: GPCR/G protein|OX Receptor Synonyms: N/A Formula: C31H38N2O5 N/A Molecular Weight: 518...

ML 289 | B5783-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: negative allosteric modulator of mGlu3 receptors Category: Neuroscience|GluR Synonyms: N/A Formula: C22H23NO3 N/A Molecular Weight: 349.42 Chemical...

VUF 11207 fumarate | B5711-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: ACKR3 (CXCR7) chemokine receptor agonist Category: GPCR/G protein|Chemokine Receptors Synonyms: N/A Formula: C27H35FN2O4·C4H4O4 N/A ...

BETP | B5710-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: glucagon-like peptide 1 (GLP-1) receptor modulator Category: GPCR/G protein|Glucagon Receptor Synonyms: N/A Formula: C20H17F3N2O2S N/A Molecular Weight:...

TC LPA5 4 | B5689-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: LPA5 receptor antagonist Category: GPCR/G protein|LPA Receptor Synonyms: N/A Formula: C23H23ClN2O3 N/A Molecular Weight: 410.89 Chemical Name: 5-...

LUF 5834 | B5653-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: A2A and A2B adenosine receptor partial agonist Category: GPCR/G protein|Adenosine Receptor Synonyms: N/A Formula: C17H12N6OS N/A Molecular Weight: ...

EMPA | B5641-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: OX2 receptor antagonist Category: GPCR/G protein|OX Receptor Synonyms: N/A Formula: C23H26N4O4S N/A Molecular Weight: 454.54 Chemical Name: N-ethyl-2-...

GPBAR-A | B5616-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: agonist of bile acid receptor GPBAR1 Category: Metabolism|Lipid Metabolism Synonyms: N/A Formula: C23H15F7N2O2 N/A Molecular Weight: 484.37 ...

TC-N 22A | B5565-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: mGlu4 receptor positive allosteric modulator Category: Neuroscience|GluR Synonyms: N/A Formula: C14H13N5S N/A Molecular Weight: 283.35 Chemical...

Ro 67-7476 | B5560-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: positive allosteric modulator of mGlu1 receptors Category: Neuroscience|GluR Synonyms: N/A Formula: C17H18FNO2S N/A Molecular Weight: 319.39 ...

AR-M 1000390 hydrochloride | B5558-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Delta-opioid receptor agonist,low-internalizing Category: Endocrinology and Hormones|Opioid Receptor Synonyms: N/A Formula: ...

PSB 0777 ammonium salt | B5557-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: adenosine A2A receptor full agonist Category: GPCR/G protein|Adenosine Receptor Synonyms: N/A Formula: C18H20N5O7S2·NH4 N/A Molecular...

GSK 9027 | B5528-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: glucocorticoid receptor agonist Category: GPCR/G protein|Glucocorticoid Receptor Synonyms: N/A Formula: C27H19F4N3O2S N/A Molecular Weight: 525.52 ...

JNJ 5207852 dihydrochloride | B5513-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: histamine H3 receptor neutral antagonist Category: Neuroscience|Histamine Receptor Synonyms: N/A Formula: C20H32N2O·2HCl N/A ...

SR 140333 | B5510-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: NK1 receptor antagonist Category: Neuroscience|Substance P/NK1 Receptor Synonyms: N/A Formula: C37H45Cl3N2O2 N/A Molecular Weight: 656.12 ...

Brain natriuretic peptide (1-32) (human) | B5442-10 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: agonist at atrial natriuretic peptide (ANP) receptor A (NRP1) Category: Others|Natriuretic Peptide Receptors Synonyms: N/A ...

ACTH (1-39) | B5434-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: melanocortin receptor 2 (MC2) agonist Category: GPCR/G protein|Melanocortin (MC) Receptors Synonyms: N/A Formula: C207H308N56O58S N/A Molecular...

GLYX 13 | B5419-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: NMDA receptor partial agonist Category: Membrane Transporter/Ion Channel|NMDA Receptor Synonyms: N/A Formula: C18H31N5O6 N/A Molecular Weight: 413.47...

NDT 9513727 | B5411-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: C5a receptor (C5aR) competitive antagonist Category: N/A Synonyms: N/A Formula: C36H35N3O4 N/A Molecular Weight: 573.68 Chemical Name: 1-...

Dynorphin B | B5390-10 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: endogenous agonist for the kappa opioid receptor Category: Endocrinology and Hormones|Opioid Receptor Synonyms: N/A Formula: C74H115N21O17 N/A ...

Neuropeptide W-23 (human) | B5361-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous peptide agonist of Neuropeptide B/Neuropeptide W receptors NPBW1 and NPBW2 Category: GPCR/G protein|Peptide Receptors Synonyms: ...

SB 258719 hydrochloride | B5334-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Selective 5-HT7 receptor antagonist Category: GPCR/G protein|5-HT Receptor Synonyms: N/A Formula: C18H30N2O2S·HCl N/A Molecular...

(+)-Igmesine hydrochloride | B5294-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: σ1 receptor ligand Category: GPCR/G protein|Sigma Receptor Synonyms: N/A Formula: C23H29N·HCl N/A Molecular Weight: 355.94 ...

MNI-caged-D-aspartate | B5286-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Agonist at NMDA receptors and EAAT substrate Category: Membrane Transporter/Ion Channel|NMDA Receptor Synonyms: N/A Formula: C13H15N3O6 N/A...

Motilin (human, porcine) | B5284-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous motilin receptor ligand Category: GPCR/G protein|Motilin Receptor Synonyms: N/A Formula: C120H188N34O35S N/A Molecular...

BAM 22P | B5155-5 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Potent endogenous agonist peptide for the newly identified sensory neuron specific receptor (SNSR); Category: Endocrinology and Hormones|Opioid Receptor ...

Astressin | B5147-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: corticotropin-releasing factor (CRF) receptor antagonist Category: GPCR/G protein|Non-selective CRF Synonyms: N/A Formula: C161H269N49O42 N/A ...

LY 288513 | B5125-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Selective CCK2 receptor antagonist Category: GPCR/G protein|CCK2 Receptors Synonyms: N/A Formula: C22H18BrN3O2 N/A Molecular Weight: 436.3 ...

Orexin B (mouse) | B5119-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous agonist at orexin receptors Category: GPCR/G protein|Orexin Synonyms: N/A Formula: C126H215N45O34S N/A Molecular Weight: 2936.40 ...

Orexin B (human) | B5118-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous agonist at orexin receptors Category: GPCR/G protein|Orexin Synonyms: N/A Formula: C123H212N44O35S N/A Molecular Weight: 2899.36 ...

Orexin A (human, rat, mouse) | B5117-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous agonist at orexin receptors Category: GPCR/G protein|Orexin Synonyms: N/A Formula: C152H247N47O44S4 N/A Molecular...

FR 139317 | B5082-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: highly potent and selective ETA endothelin receptor antagonist Category: GPCR/G protein|ETA Receptors Synonyms: N/A Formula: C33H44N6O5 N/A ...

CGRP 8-37 (human) | B5073-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Peptide antagonist for CGRP1 receptors Category: GPCR/G protein|Calcitonin and Related Receptors Synonyms: N/A Formula: C139H230N44O38 N/A ...

Endothelin 3 (human, rat) | B5062-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous neuropeptide with selectivity for the putative ETC endothelin receptor Category: GPCR/G protein|Endothelin Receptor Synonyms: N/A...

Pancreatic Polypeptide (human) | B5060-5 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous high affinity agonist for human NPY Y4 receptor Category: GPCR/G protein|NPY Receptors Synonyms: N/A Formula: ...

Nociceptin | B5033-25 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: Endogenous ligand for the NOP opioid receptor Category: GPCR/G protein|NOP Receptor Synonyms: N/A Formula: C79H129N27O22 N/A Molecular Weight: 1809...

MRS 2179 tetrasodium salt | B5032-50 | Gentaur US, UK & Europe Disrtribition Purity: N/A Short Sumary: competitive antagonist at P2Y1 receptors Category: GPCR/G protein|P2Y Receptor Synonyms: N/A Formula: C11H13N5O9P2Na4 N/A Molecular...

JNJ-31020028 | B4827-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: selective brain penetrant antagonist of neuropeptide Y2 receptor Category: Neuroscience|Neuroscience Peptides Synonyms: N/A Formula: C34H36FN5O2 ...

AL 8810 | B4575-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Antagonist of prostaglandin F2α (FP) receptor. Category: GPCR/G protein|Prostaglandin Receptor Synonyms: N/A Formula: C24H31FO4 N/A Molecular Weight: ...

DDR1-IN-1 | B3383-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: selective DDR1 receptor tyrosine kinase inhibitor Category: Tyrosine Kinase|DDR1/DDR2 Receptor Synonyms: N/A Formula: C30H31F3N4O3 N/A Molecular...

ACT-132577 | B3279-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: ETA/ETB receptors antagonist Category: N/A Synonyms: N/A Formula: C16H14Br2N6O4S N/A Molecular Weight: 546.19 Chemical Name: N/A CAS: ...

Doxercalciferol | B2091-500 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Vitamin D receptor activator Category: Vitamin D Related|VD/VDR Synonyms: N/A Formula: C28H44O2 N/A Molecular Weight: 412.66 Chemical...

MK-3207 HCl | B1436-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Potent CGRP receptor antagonist Category: N/A Synonyms: N/A Formula: C31H30ClF2N5O3 N/A Molecular Weight: 594.05 Chemical Name: 2-[ (8R)-8-...

Rimonabant | B1429-1000 | Gentaur US, UK & Europe Disrtribition Purity: 0.9816 Short Sumary: CB1 receptor antagonist Category: GPCR/G protein|Cannabinoid Receptor Synonyms: N/A Formula: C22H21Cl3N4O N/A Molecular Weight: 463.79 ...

Siramesine | B1297-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Sigma (σ) receptor agonist Category: GPCR/G protein|Sigma Receptor Synonyms: N/A Formula: C30H31FN2O N/A Molecular Weight: 454.58 Chemical...

TGR5 Receptor Agonist | B1185-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.998 Short Sumary: TGR5 G-protein receptor agonist Category: Others|Others Synonyms: N/A Formula: C18H14Cl2N2O2 N/A Molecular Weight: 361.22 Chemical...

Palovarotene | B1175-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.9841 Short Sumary: Selective retinoic acid receptor gamma (RAR-γ) agonist Category: Others|RAR/RXR Synonyms: N/A Formula: C27H30N2O2 N/A Molecular Weight: 414...

GSK962040 | B1149-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Motilin receptor agonist Category: Others|Others Synonyms: N/A Formula: C25H33FN4O N/A Molecular Weight: 424.55 Chemical Name: 1-[4-...

GSK962040 hydrochloride | B1137-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Small molecule, selective motilin receptor agonist Category: GPCR/G protein|Motilin Receptor Synonyms: N/A Formula: C25H34ClFN4O N/A ...

Tarafenacin D-tartrate | B1133-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Highly selective M3 muscarinic receptor antagonist Category: Neuroscience|AChR Synonyms: N/A Formula: C25H26F4N2O8 N/A Molecular...

Tarafenacin | B1132-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: M3 muscarinic receptor antagonist Category: Neuroscience|AChR Synonyms: N/A Formula: C21H20F4N2O2 N/A Molecular Weight: 408.39 Chemical Name: ...

MDL-29951 | B1038-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Glycine antagonist of NMDA receptor activation Category: Membrane Transporter/Ion Channel|NMDA Receptor Synonyms: N/A Formula: C12H9Cl2NO4 N/A ...

SR1078 | A3835-200 | Gentaur US, UK & Europe Disrtribition Purity: 0.9865 Short Sumary: Orphan receptor agonist Category: Tyrosine Kinase|ROR Synonyms: SR 1078;SR-1078 Formula: C17H10F9NO2 SR 1078;SR-1078 Molecular Weight: 431.25 ...

Rimonabant hydrochloride | A3766-1000 | Gentaur US, UK & Europe Disrtribition Purity: 0.9801 Short Sumary: CB1 receptor inverse agonist Category: GPCR/G protein|Cannabinoid Receptor Synonyms: SR 141716A; SR 151716A Formula: C22H22Cl4N4O ...

MK-2894 | A3613-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: EP4 receptor inhibitor Category: GPCR/G protein|EP4 Receptor Synonyms: MK 2894;MK2894 Formula: C25H22F3NO3S MK 2894;MK2894 Molecular Weight: 473.51 ...

MK-0974 | A3612-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: CGRP receptor antagonist Category: Neuroscience|CGRP Synonyms: Telcagepant;MK0974;MK 0974 Formula: C26H27F5N6O3 Telcagepant;MK0974;MK 0974 Molecular...

Metiamide | A3598-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Histamine H2-receptor antagonist Category: Others|Others Synonyms: N/A Formula: C9H16N4S2 N/A Molecular Weight: 244.38 Chemical Name: ...

glucagon receptor antagonists 1 | A3435-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Glucagon receptor antagonist,highly potent Category: GPCR/G protein|Glucagon Receptor Synonyms: glucagon receptor antagonists-1 ...

Ercalcidiol | A3395-25 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Vitamin D2 metabolite,ligand of VDR-like receptors Category: Vitamin D Related|VD/VDR Synonyms: 25-hydroxy Vitamin D2 Formula: C28H44O2 25-hydroxy...

Capadenoson | A3277-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Adenosine A1 receptor agonist Category: GPCR/G protein|Adenosine Deaminase#Metabolism|Adenosine Deaminase Synonyms: BAY 68-4986 Formula: ...

Capadenoson | A3277-50 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: Adenosine A1 receptor agonist Category: GPCR/G protein|Adenosine Deaminase#Metabolism|Adenosine Deaminase Synonyms: BAY 68-4986 Formula: ...

Alvimopan dihydrate | A3163-500 | Gentaur US, UK & Europe Disrtribition Purity: 0.98 Short Sumary: μ-opioid receptor antagonist,peripherally acting Category: Endocrinology and Hormones|Opioid Receptor Synonyms: LY 246736 dihydrate;ADL 8-2698...

Ramelteon | A1748-100 | Gentaur US, UK & Europe Disrtribition Purity: 0.9989 Short Sumary: Agonist of melatonin receptor (M1-M2),highly selective Category: GPCR/G protein|MT Receptor Synonyms: N/A Formula: C16H21NO2 N/A Molecular...