K252a | 27033

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SKU:
412-27033
€618.00
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Description

K252a | 27033 | Gentaur US, UK & Europe Disrtribition

Category: Kinase/Kinase Inhibitors

Application: N/A

Background: N/A

Description: K252a is a general kinase inhibitor that inhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), PKG (Ki = 20 nM), CaMK (Ki = 1.8 nM), and phosphorylase kinase (IC50 = 1.7 nM). It functions by acting competitively with ATP and noncompetitively with the substrate.

Product Type: Inhibitor

Shippement Condition: -20°C

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